ISSN (Print):
2949-6810
ISSN (Online):
2949-6829

Drug Metabolism and Bioanalysis Letters

All Open Access articles of this journal are also available on ScienceDirect.

(Formerly Drug Metabolism Letters) (Continued as Drug Metabolism and Bioanalysis)

Indexed in: Scopus, MEDLINE/PubMed, Cabell's Directory/Journalytics... View all

Volume 18 , Issues 2, 2025


Aims & Scope

Drug Metabolism and Bioanalysis Letters is an interdisciplinary, peer-reviewed journal that publishes letters, original research papers, mini-reviews, and guest-edited issues in all important aspects of drug metabolism, pharmacokinetics, and bioanalysis.

The scope includes in vitro systems, including CYP-450; enzyme induction and inhibition; drug-drug interactions and enzyme kinetics; pharmacokinetics, toxicokinetics, species scaling and extrapolations; P-glycoprotein and transport carriers; target organ toxicity and interindividual variability; drug metabolism and disposition studies; extrahepatic metabolism; phase I and phase II metabolism; bioactivation; recent developments for the identification of drug metabolites, reactive intermediate, and glutathione conjugates.

Additionally, LC/MS and other key detection methods, including ligand binding assays, sample preparation, chromatography and separation sciences, and method development and validation, are included, with applications in drug and metabolite assays, pharmacokinetic/toxicokinetic assays, biomarker assays, immunogenicity assays, diagnostic assays. Topics covered in this interdisciplinary journal include:

  1. Analytical Method and Drug Metabolism
  2. Bioavailability and Biopharmacy
  3. Cytochrome 450 Drug Metabolism
  4. Cytotoxicity
  5. Drug Absorption and Disposition
  6. Drug Biotransformation
  7. Drug Delivery System
  8. Drug-Drug Interaction
  9. Drug Food Interaction
  10. Drug Metabolizing Enzymes
  11. Drug Toxicology
  12. Drug Transporters
  13. Drugs and CYP2D6
  14. Factors Affecting Drug Metabolism
  15. Hepatic Metabolism of Drugs
  16. P-Glycoprotein and Transport Carriers
  17. Pharmacokinetics and Pharmacodynamics
  18. Phase I and II Drug Metabolism
  19. Reactive Metabolites
  20. Therapeutic Drug Monitoring
  21. Xenobiotics

Drug Metabolism and Bioanalysis Letters is an international, peer-reviewed journal on all aspects of drug metabolism and bioanalysis published half-yearly (print & online) by Bentham Science Publishers.

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