Upcoming Articles of Medicinal Chemistry:
Contents
Four-Component Synthesis of 1,2-Dihydropyridine Derivatives and their Evaluation as Anticancer Agents
Mohamed A. O. Abdelf-Fattah, Mahmoud A. M. El-Naggar, Rasha M. H. Rashied, Bernard D. Gary, Gary A. Piazza and Ashraf H. Abadi
CoMFA and CoMSIA Studies of 1,2-Dihydropyridine Derivatives as Anticancer Agents
Ismail Salama, Mohamed A. O. Abdel-Fattah, Marwa S. Hany, Shaimaa A. El-Sharif, Mahmoud A. M. El-Naggar, Rasha M. H. Rashied, Gary A. Piazza and Ashraf H. Abadi
First Study on Antimicriobial Activity And Synergy between Isothiocyanates And Antibiotics Against Selected Gram-Negative And Gram-Positive Pathogenic Bacteria From Clinical And Animal Source
Carla Dias, Alfredo Aires, Richard N. Bennett, Eduardo A. S. Rosa and Maria J. Saavedra
In vitro Anti-glycation and Anti-oxidant Properties of Synthesized Schiff Bases
Sabina Jhaumeer-Laulloo, Minu Gupta Bhowon, Shabneez Mungur, Mohamad Fawzi Mahomoodally and Anwar Hussein Subratty
Synthesis and Biological Evaluation Of The Salicylamide and Salicylic Acid Derivatives As Anti-Estrogen Agents
Yasemin Dündar, Yasemin Özatik, Orhan Özatik, Volkan Ergin, Tijen Önkol, Adnan Menevşe, Kevser Erol and M. Fethi Şahin
Synthesis and Activity of [{Cis-PtCl(NH3)2}2µ{Trans-Pt(3-Hydroxypyridine)2(H2N(CH2)6NH2)2}]Cl4 in the Human Ovarian Tumour Models
Shahnaz AH Hamad, Philip Beale, Jun Qing Yu, Keith Fisher and Fazlul Huq
Biological and Anti-inflammatory Evaluation of Two Thiazole Compounds in RAW Cell Line: Potential Cyclooxygenase-2 Specific Inhibitors
Eva Hamade, Aida Habib, Ali Hachem, Alaa H. Hussein, Malak Abbas, Taghreed Hirz, Mirvat Al Masri and Wissam H. Faour
New Adamantane Derivatives with Sigma Affinity and Antiproliferative Activity
Stefanos Riganas, Ioannis Papanastasiou, George B. Foscolos, Andrew Tsotinis, Kostas Dimas, Vassilios N. Kourafalos, Andreas Eleutheriades, Vassilios I. Moutsos, Humaira Khan, Prassa Margarita, Stavroula Georgakopoulou, Angeliki Zaniou, Maria Theodoropoulou, Athanasios Mantelas, Stavroula Pondiki and Alexandre Vamvakides
Synthesis of Novel 4-Aryl-1,2,3,4-tetrahydroisoquinolines as Probes for Dopamine Receptor Ligands
Gianfabio Giorgioni, Dario Ambrosini, Giovanni Filippo Palmieri, Barbara Costa, Antonio Di Stefano and Claudia Martini
A Quantitative Structure-Activity Relationship Study on a Few Series of Anti-hepatitis C Virus Agents
Jonish Varshney, Anjana Sharma and Satya P. Gupta
Synthesis and Antiglycation Activity of Kaempferol-3-O-rutinoside (Nicotiflorin)
Sajan Lal Shyaula, Ghulam Abbas, Hina Siddiqui, Samina A. Sattar, M. Iqbal Choudhary and Fatima Z. Basha
Synthesis and β-Glucuronidase Inhibitory Potential of Benzimidazole Derivatives
Khalid Mohammed Khan, Momin Khan, Nida Ambreen, Fazal Rahim, Shagufta Naureen, Shahnaz Perveen, M. Iqbal Choudhary and Wolfgang Voelter
Synthesis and Biological Evaluation of Some New N4-Aryl Substituted 5-Chloroisatin-3 thiosemicarbazones
Humayun Pervez, Muhammad Ramzan, Muhammad Yaqub, Faiz-Ul-Hassan Nasim and Khalid Mohammed Khan
2,4,6-Trichlorophenylhydrazine Schiff Bases as DPPH Radical and Super Oxide Anion Scavengers
Khalid Mohammed Khan, Zarbad Shah, Viqar Uddin Ahmad, Momin Khan, Muhammad Taha, Fazal Rahim, Sajjad Ali, Nida Ambreen, Shahnaz Perveen, M. Iqbal Choudhary andWolfgang Voelter
Application of Artificial Neural Networks for the Prediction Of Antitumor Activity of A Series of Acridinone Derivatives
Marcin Koba
Synthesis and Biological Evaluation of 3΄-C-Ethynyl and 3΄-C-(1,4-disubstituted-1,2,3-triazolo) Double-Headed Pyranonucleosides
Christos Kiritsis, Stella Manta, Ioannis Papasotiriou, Evdoxia Coutouli-Argyropoulou, Sakellarios Trakossas, Jan Balzarini and Dimitri Komiotis
Structure-Activity Relationships of Pyrrole Hydrazones as New Anti-Tuberculosis Agents
Iglika Lessigiarska, Ilza Pajeva, Penka Prodanova, Maya Georgieva and Atanas Bijev
S-Ntrosylation and Attenuation of Excessive Calcium Flux by Pentacycloundecane Deriva Tives
Hendrik, J.R. Lemmer, Jacques Joubert, Sandra van Dyk, Francois, H. van der Westhuizen and Sarel, F. Malan
Serum Specific Vasopressin-Degrading Activity is Related to Blood Total Cholesterol Levels in Men But not In Women
Ramírez-Expósito María Jesús, Arrazola Marcelina, Carrera- González María Pilar, Arias de Saavedra José Manuel, Sánchez-Agesta Rafael, Mayas María Dolores and Martínez-Martos José Manuel
SAR Analysis of New Dual Targeting Fluoroquinolones. Implications of the Benzenesulfonyl Group
Marcelo J. Nieto, Adriana B. Pierini, Nidhi Singh, Christopher R. McCurdy, Ruben H. Manzo and María R. Mazzieri
Prodrug Strategies in Ocular Drug Delivery
Megha Barot, Mahuya Bagui, Mitan R. Gokulgandhi and Ashim K. Mitra
Synthesis and Biological Evaluation of Naloxone and Naltrexone-Derived Hybrid Opioids
Bahman E. Nassim and Ming-Lei Wang
A QSAR Analysis of 2-phenoxy-N-substituted acetamide Analogues as Hypoxia-Inducible Factor-1(HIF-1) inhibitors: A Rational Approach to Anticancer Drug Design
Malleshappa N. Noolvi, Harun M. Patel and Sarita Kamboj
Synthesis, In Vitro And In Silico Ns5b Polymerase Inhibitory Activity Of Benzimidazole Derivatives
Vaishali M. Patil, Gurukumar K. R., Maksim Chudayeu, Satya Prakash Gupta, Subeer Samanta, Neeraj Masand and Neerja Kaushik-Basu
A new Class of Anticonvulsants Possessing 6 Hz Psychomotor Seizure Test Activity: 2-(1H-Benzotriazol-1-yl)-N'-[Substituted] Acetohydrazides
Praveen Kumar, Birendra Shrivastava, Surendra Nath Pandeya, Laxmi Tripathi and James P. Stables
Synthesis and Biological Evaluation of a Series of 6,7-dimethoxy-1-(3,4-dimethoxybenzyl)-2-substituted Tetrahydroisoquinoline Derivatives
Zhi-hong Zou, Xiao-bu Lan, Chun-lei Tang, Xiao-yun Zhu, Bao-min Liu, Hai Qian, Wen-long Huang and Yun-man Li
Generation of Pharmacophore and Atom Based 3D-QSAR Model of Novel Isoquinolin-1-one and Quinazolin-4-one-type Inhibitors of TNFα
Pradeep Hanumanthappa, Mahesh K. Teli and Rajanikant G. Krishnamurthy
A QSAR Study of Biphenyl Analogues of 2-Nitroimidazo-[2, 1-b] [1, 3] - oxazines as Antitubercular Agents using Genetic Function Approximation
Supratim Ray and Partha Pratim Roy
Differences in Vanadocene Dichloride And Cisplatin Effect on MOLT-4 Leukemia and Human peripheral Blood Mononuclear Cells
Havelek Radim, Siman Pavel, Cmielova Jana, Stoklasova Alena, Vavrova Jirina, Vinklarek Jaromir, Knizek Jiri and Rezacova Martina
In Vitro Synergy Testing of Anidulafungin with Fluconazole, Tioconazole, 5-Flucytosine and Amphotericin B Against Some Candida spp
Antonio Rosato, Monica Piarulli, Brigida Immacolata Pia Schiavone, Maria Teresa Montagna, Giuseppina Caggiano, Marilena Muraglia, Addolorata Carone, Carlo Franchini and Filomena Corbo
Structural Insight for Imidazopyridazines as Malarial Kinase PfPK7 Inhibitors Using QSAR Techniques
Nitendra K. Sahu and D. V. Kohli
Substituted Urea Derivatives: A Potent Class of Antidepressant Agents
Shahnaz Perveen, Sana Mustafa, Muhammad A. Khan, Ahsana Dar Khalid M. Khan and Wolfgang Voelter
A QSAR Study on Novel Series of Carbonic Anhydrase Inhibitors hCA IX—Tumor-Associated (Hypoxia)
Shalini Singh
Synthesis and 188Re Radiolabelling of Dendrimer Polyamide Amine (PAMAM) Folic Acid Conjugate
Wei Cui, Yuanqing Zhang, Xiaoping Xu and Yu-Mei Shen
Computational Approaches To Improve Aggrecanase-1 Inhibitory Activity Of (4-Keto) Phenoxy) Methyl biphenyl-4-Sulfonamide: Group Based QSAR and Docking Studie
Ponnurengam Malliappan Sivakumar, J. Mohanapriya, Naga Vignesh Selva Raj, G. Ramesh and Mukesh Doble
In vitro Antibacterial and Antifungal Activity of Salicylanilide Pyrazine-2-Carboxylates
Martin Krátký, Jarmila Vinšová and Vladimír Buchta
Design, Synthesis and Multidrug Resistance Reversal Activity Evaluation of 8-Oxocoptisine Derivatives
Jian Bo Wu, Fan Lei, Xiang Juan Cui, Yun He, Li Hai, Juan Zhang and Yong Wu
Design, Synthesis and Antiproliferative Studies Of 2-Acetylamino-Thiazole-5-Carboxamide Derivatives
Wukun Liu, Jinpei Zhou, Yu Zheng, Fan Qi, Huibin Zhang, Hai Qian, Jing Wang, Yanhua Chen and Ronald Gust
Synthesis of 3-(2, 8, 9-Trioxa-5-Aza-1-Germatricyclo [3.3.3.0] Undecane-1-Yl)-3-(4-Hydroxyl-3- Methoxyphenyl)-Propionic Acid and its Inhibitory Effect on the Cervical Tumor U14 In Vitro and In Vivo
Lianbao Ye, Xiaomin Ou, Xuedong Peng and Yan Luo
A QSAR Study on a Series of Pyrrole Derivatives Acting as Lymphocyte-Specific Kinase (Lck) Inhibitors
Zaihra Anwe and Satya P. Gupta
Acylhydrazide Schiff Bases: DPPH Radical and Superoxide Anion Scavengers
Khalid Mohammed Khan, Muhammad Taha, Farzana Naz, Salman Siddiqui, Sajjad Ali, Fazal Rahim, Shahnaz Perveen and M. Iqbal Choudhary
The Preformulation Stability Studies of a Proline Prodrug of Methotrexate
Ann Stephenson, Zhiqian Wu and Xudong Yuan
Synthesis of a Biodegradable Magnetic Nanomedicine Based on the Antitumor Molecule Tegafur
José L. Arias, Eva Sáez-Fernández, Margarita López-Viota, Rafael A. Biedma-Ortiz and M Adolfina Ruiz
Monodisperse Nanoparticles from Self-Assembled Amphiphilic Cyclodextrins: Modulable Tools for the Encapsulation and Controlled Release of Pharmaceuticals
Alejandro Mendez-Ardoy, Marta Gómez-García, Annabelle Gèze, Jean-Luc Putaux, Denis Wouessidjewe, Carmen Ortiz Mellet, Jacques Defaye, José M. García Fernández and Juan M. Benito
Use of Flow Focusing® Technology to Produce Tobramycin-Loaded Plga Microparticles for Pulmonary Drug Delivery
L. Martín-Banderas, M.A. Holgado, J. Álvarez-Fuentes and M. Fernández-Arévalo
Preparation, Chemical and Electrical Characterizations of Lipid Nanoparticles Loaded with Dihydroxybenzophenone
Hierrezuelo Jesús, Benavente Juana, López–Romero Juan Manuel, Martínez de Yuso Maria del Valle and Rodríguez–Castellón Enrique
Diagnosis of Alterations of Serum Calcium Metabolism
F. Lumachi, P. Cappelletti, R. Tozzoli, S.M.M. Basso, G. Luisetto and V. Camozzi
Treatment of Acute Hypercalcemia
S.M.M. Basso, F. Lumachi, F. Nascimben, G. Luisetto and V. Camozzi
Treatment of Chronic Hypercalcemia
V. Camozzi, G. Luisetto, S.M.M. Basso, P. Cappelletti, R. Tozzoli and F. Lumachi
|
