ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 13, 10 Issues, 2016


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Letters in Drug Design & Discovery

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Editor-in-Chief:
Atta-ur-Rahman, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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Upcoming Articles (E-Pub Abstracts ahead of Print)

Quinoline derivatives as novel depigmenting and antioxidant agents


Rebeca Mól Lima, Jordana de Abreu Lazzarini, Isabela Oliveira Souza, Adilson David Silva, Nádia Rezende Barbosa Raposo and Kauana Cristina de Souza.


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Synthesis and nematocidal activity of novel pyrazole carboxamide derivatives against Meloidogyne incognita


Xing-Hai Liu.


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3D-QSAR, molecular docking and molecular dynamics studies of 2,4-diarylaminopyrimidine analogues (DAAP analogues) as potent ALK inhibitors


Fu long Wu, Qian qian Lv, Zhong hua Wang, Dan dan Li, Peng Peng, Yan Yin, Si heng Cui and Fan hong Wu.


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Design, Synthesis and Biological Evaluation of Amino-Pyrazole Derivatives


Chunqi Hu, Jianfeng Shen and Wenting Du.


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Anti-biofilm and antibacterial effects of novel metal-coordinated sulfamethoxazole against Escherichia coli.


Caren Rigon Mizdal, Sílvio Terra Stefanello, Pauline Cordenonsi Bonez, Vanessa Albertina Agertt, Vanessa da Costa Flores, Grazielle Guidolin Rossi, Fallon dos Santos Siqueira, Lenice de Lourenço Marques and Marli Matiko Anraku Campos.


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Combined 3D-QSAR, Pharmacophore and Docking Studies on Benzenesulfonamide Derivatives as Potent 12-Lipoxygenase Inhibitors


Chunhong An, Mao Shu, Xiaoli Zai, Zichao Chang, Yong Hu and Zhihua Lin.


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In Vivo Antimalarial and In Vitro Antileishmanial Activity of 4-Aminoquinoline Derivatives Hybridized to Isoniazid or Sulfa or Hydrazine Groups


Clarice Abramo, Roberta R. Soares, Luciana MR Antinarelli, Isabela de Oliveira Souza, Fernanda V. Lopes, Kézia Katiani Gorza Scopel and Adilson D da Silva.


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NF-kappaB Inhibitors in Head and Neck Cancer


Siddavaram Nagini, Kranthi Kiran Kishore Tanagala and Indranil Chattopadhyay.


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Synthesis of New Benzofuran-Pyrazole Hybrids as Potential Antibiofilm Agents


Gejjalagere S Lingaraju, Somashekaraiah Rakesh, Koravangala S Vinay Kumar, Kanchepalli Poornachandra Rao, Marikunte Y Sreenivasa and Maralinganadoddi P Sadashiva.


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Synthesis of Novel 4-(Dimethylaminoalkyl)piperazine-1-carbodithioate Derivatives as Cholinesterase Inhibitors


Ulviye Acar, Serkan Levent, Begüm Nurpelin Sağlık, Yusuf Özkay and Zafer Asım Kaplancıklı.


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Sequential Therapy For Helicobacter Pylori In Elderly Patients: Effectiveness, Safety And Predictors Of Success


Giuseppe Losurdo, Andrea Iannone, Floriana Giorgio, Michele Barone, Mariabeatrice Principi, Enzo Ierardi and Alfredo Di Leo.


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Molecular mechanisms and potential treatment targets for ovarian cancer by analyzing transcriptional regulatory network


Fei Wu, Xinrui Liu, Yujie Sui, Tianmin Xu and Manhua Cui.


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Pentoxifylline alleviates proteinuria in fructose model of metabolic syndrome


Hany M. El-Bassossy, Basma Eid and Ahmad Azhar.


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Relationships between the structural properties of flavonoids and their inhibitory activities against matrix metallopeptidase 9


Soon Young Shin, Hyeryoung Jung, Yearam Jung, Beom Soo Kim, Young Han Lee and Yoongho Lim.


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Identification of thiazoloquin(az)olin(on)es derivatives as CD38 inhibitors through structure-activity relationships and molecular docking simulations


Xiaodong Gao and Jie Yu Ren.


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Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches


Sk. Abdul Amin, Nilanjan Adhikari, Ramkishore Agrawal, Tarun Jha and Shovanlal Gayen.


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Novel Second Generation HIV Integrase Inhibitor- DOLUTEGRAVIR : an emerging weapon against HIV


Vivek Jain, Diksha Gupta, Ashutosh Pareek and Yashumati Ratan Bhardwaj.


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3D-QSAR studies of novel cytotoxic bufadienolides via CoMFA and CoMSIA approaches


Jian Jie, Hui Lin, Kangjia Liu, Yushui Han, Jialiang Guo, Longxin Lin, Yiqun Chang, Gaokeng Xiao, Weimin Chen and Pinghua Sun.


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Caffeic Acid Phenethyl Ester Restores Adipocyte Function Following Lipopolysaccharide treatment


Ignazio Barbagallo, Giovanni Li Volti, Valeria Sorrenti, Claudia Di Giacomo, Rosaria Acquaviva, Marco Raffaele, Fabio Galvano and Luca Vanella.


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Improved Anti-inflammatory Activity and Potential Cytoprotective Properties of Tolfenamic Acid, Naproxen and Indomethacin Derivatives


Panagiotis Theodosis-Nobelos, Theodora C Politou, Chrysoula Athanasekou and Eleni A Rekka.


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Computational Analysis of Pyridopyrimidine-based Polo Like Kinase 2 (PLK2) Inhibitors: Probing the Relationship between Structural Features and Anticancer Potency


Anand Balupuri, Pavithra K. Balasubramanian and Seung Joo Cho.


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Design, synthesis and antidepressant and anticonvulsant effect of 1-alkoxy -1H-benzo[d][1,2,3]triazole derivatives


Qinghao Jin, yingchun quan, yan han, di yu, qiuping dai and zhoujun zheng.


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Fe3+-Tryptophan-3-Hydroxy-2-Methyl or ethyl pyridinones Towards Novel Molecular Tumor Nuclear Resonance Imaging Agents


Ali Khalaj, Shadi Hosseini, Rahimeh Rasouli, Artin Assadi, Seyedeh Ghoreishi and Mehdi Shafiee Ardestani.


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