ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 14, 12 Issues, 2017


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Letters in Drug Design & Discovery

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Editor-in-Chief:
G. Perry
University of Texas
San Antonio, TX
USA


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Abstracts Ahead of Print

Synthesis and antioxidant evaluation of a new class of thienopyrimidine-rhodanine hybrids


Kerru Nagaraju , Venkata H.S.S. Bhaskaruni, Ravada Kishore , Suresh Maddila, Parvesh Singh and Jonnalagadda B Sreekantha.


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Nalidixic Acid Schiff bases: Synthesis and Biological Evaluation


Asif Husain, Munendra Mohan Varshney, Versha Parcha, Aftab Ahmad and Shahalam Khan.


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Nalidixic Acid Schiff bases: Synthesis and Biological Evaluation


Asif Husain, Munendra Mohan Varshney, Versha Parcha, Aftab Ahmad and Shahalam Khan.


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Novel 11,12H-dihydronaphthalene[1,2-b]quinoline as Atypical Antipsychotic


Maria Matilde Ramirez Moran, Jorge Eduardo Angel, Natividad Herrera Cano, Biagina Del Carmen Migliore, Rodolfo Izquierdo, Jaime Charris, Simón López, Anita Israel, Ana Santiago, Roberto Ross, Luis Perdomo, Akram Samear Dabian, Mariagracia Vera, Alejandra Villalba and Ligia Biagina Angel Migliore.


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Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors


Gülhan Turan-Zitouni, Weiam Hussein, Begüm Nurpelin Sağlık, Merve Baysal and Zafer Asım Kaplancıklı.


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Design, synthesis and biological evaluation of some novel thiazole-2-carboxamide derivatives as antitumor agents


Haibo Wang, Zhengjiang Cai, Shan Zheng, Huidan Ma, Haiming Lin and Xiaohe Zheng.


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Synthesis, biological evaluation, molecular docking study and acute oral toxicity study of coupled Imidazolyl-Pyrimidine derivatives


Shailee V. Tiwari, Anna Pratima G. Nikalje, Deepak K. Lokwani, Aniket P. Sarkate and Kizukala Jamir.


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A Comprehensive Review on Recent Developments in the Field of Biological Applications of Potent Pyrazolines Derived from Chalcone Precursors


Vinutha V. Salian, Badiadka Narayana, Balladka K. Sarojini and Kullaiah Byrappa.


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A Comprehensive Review on Recent Developments in the Field of Biological Applications of Potent Pyrazolines Derived from Chalcone Precursors


Badiadka Narayana, Vinutha V. Salian, Balladka K. Sarojini and Kullaiah Byrappa.


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The antiviral effects of harmine against BoHV-1 infection in vitro


Xinyi Jiang, Jie Zou, Yuncheng Zhuang, Weifeng Yuan, Liqian Zhu and Guoqiang Zhu.


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Anti-MRSA (Multidrug resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins


Uzma Salar, Khalid Mohammed Khan, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah , Shahnaz Perveen and M Iqbal Choudhary.


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Molecular Docking Studies of Novel Thiosemicarbazone-Based Indoles as Potential PI3Kα Inhibitors


Dima A. Sabbah and Kamal Sweidan.


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Synthesis and evaluation of the anticonvulsant activities of new 5-substitued-[1,2,4]triazolo[4,3-a]quinoxalin-4(5H)-one derivatives


Guo-Rui Zhang, Yang Ren, Xiu-Mei Yin and Zhe-Shan Quan.


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Synthesis and antimicrobial activity of some new N-(1H-benzimidazol-2-yl)-2-mercaptoacetamide derivatives


Asaf Evrim Evren, Sinem Tekinkoca and Leyla Yurttas.


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Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents


Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao , Do Nguyet Que , Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han , Nguyen Thi Thuan and Nguyen-Hai Nam.


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The effectiveness of different treatment modalities for the management of ocular injuries following sulfur mustard exposure: A review


Yunes Panahi, Mostafa Naderi, Shahbaz Nekoozadeh, Seyyed Mahdi Rajaee and Amirhossein Sahebkar.


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Synthesis and Anti-oxidant Evaluation of Some Novel Sulfa Drugs


Moustafa Ahmed Gouda and Belal Hussein M Hussein.


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Design, Synthesis and In silico studies of new 5-substituted-2-(2-(5-aryl-1H-1,2,4-triazole-3-ylthio) acetyl) hydrazine carbothioamide/ carboxamides for anticonvulsant activity


Sarangapani Manda, Venkatesham Akena, Ajitha Makula and Radhika Chelamalla.


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QSAR and Molecular Docking Studies on a Series of 1-Amino-5H-pyrido [4, 3-b]indol-4-carboxamides acting as Janus Kinase 2 (JAK2) Inhibitors


K. Anita, Tabassum Zafar, Satya P. Gupta and Bashirulla Shaik.


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High throughput screening and molecular docking of calmodulin with antagonists of Trifluoperazine and Phenothiazine chemical class


Abdelmonem Messaoudi, Zarrin Basharat and Asif Naqvi.


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An Improved Preparation of (R)-3-Aminobutanol, a Key Intermediate for the Synthesis of Dolutegravir Sodium


Y. Srinivasa Rao, B. Hari Babu, I. Aminual, D. Nageshwar and PVV Satyanarayana.


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a-Glucosidase inhibition, antioxidant and docking studies of hydroxycoumarins and their mono and bis O-alkylated/acetylated analogs


Parvesh Singh, Nomandla Ngcoya, Ramgopal Mopuri, Nagaraju Kerru, Neha Manhas, Oluwakemi Ebenezer and Md Shahidul Islam.


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Microwave-assisted Synthesis and Antifungal Activity of Novel 1,2,4- Triazole Thioether Derivatives Containing Pyrimidine Moiety


Meng Xu, Ya-Bo Zhu, Mei Wang, Ikhlas A. Khan, Xing-Hai Liu and Jian-Quan Weng.


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Spices chemoconstituents as persuasive inhibitor of S. typhimurium virulent protein L-Asparaginase


Archana Vimal and Awanish Kumar.


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Pd/C-catalyzed synthesis of 4-biaryl substituted 2-amino benzo[h]chromene derivatives as potential cytotoxic agents


Meda Haritha, Chekuri Sharmila Rani, Mandava V. Basaveswara Rao and Manojit Pal.


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Synthesis and preliminarily cytotoxicity to A549, HCT116 and MCF-7 cell lines of thieno[2,3-d]pyrimidine derivatives containing isoxazole moiety


Jianping Yong, Canzhong Lu and Xiaoyuan Wu.


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