Home Page ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 11, 10 Issues, 2014


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Letters in Drug Design & Discovery

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  • 55th of 59 in

    Chemistry, Medicinal


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Editor-in-Chief:

Atta-ur-Rahman

, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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"Letters in Drug Design & Discovery should be available in every library in the pharmaceutical industry and in universities."

R. F. Borne, Associate Director
Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

Authors' Comments
I am very happy to work with editors of Bentham Science Publishers, their efficient work and good service has left a great impression on me. I hope to get the opportunity to work with Bentham Science Publishers again.

Prof. Jianhua Xu
Has contributed: Synthesis and Evaluation of 4-arylmethyl Curcumin Analgues as Potent Hsp90 Inhibitors

Letters in Drug Design & Discovery

,

Volume 11

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Number 7



Synthesis and Anticancer Activity of 2,4,5-triaryl Imidazole Derivatives

; Pp: 840 - 843

Fatemeh Elahian, Morteza Akbari, Maryam Ghasemi, Neda Behtooee, Mohaddeseh Taheri and Mohsen Amini


DOI: 10.2174/1570180811666140313233659


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Synthesis and Cholinesterase Inhibition Activity of new Pyrrolopyrimidine Derivatives


Rangaswamy Roopashree, Toreshettahally Ramesh Swaroop, Swamy Jagadish, Chakrabhavi Dhananjaya Mohan and Kanchugarakoppal Subbegowda Rangappa


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Synthesis and Antifungal Activity of 1, 3, 4-Thiadiazole Derivatives Containing Pyridine Group


Lin-Jiong Zhang, Ming-Yan Yang, Zhao-Hui Sun, Cheng-Xia Tan, Jian-Quan Weng, Hong-Ke Wu and Xing-Hai Liu


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Synthesis and in Vitro Evaluation of Thiadiazole Derivatives as AChE, BuChE and LOX Inhibitors


Mehlika Dilek Altintop, Ahmet Özdemir, Usama Abu Mohsen, Halide Edip Temel, Gülşen Akalın Çiftçi and Zafer Asim Kaplancikli


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Evaluation of Alkylating and Intercalating Properties of Mannich Bases for Cytotoxic Activity


Huseyin Istanbullu, Yalcin Erzurumlu, Petek Ballar Kirmizibayrak and Ercin Erciyas


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Theoretical Modelling of Potential Chk1 Inhibitors


Pedro M.M. Araújo, Luís Pinto da Silva and Joaquim C.G. Esteves da Silva


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Design, Synthesis and Biological Evaluation of Benzimidazole-Pyridine-Piperidine Hybrids as a new class of potent Antimicrobial Agents


Kothapally Beulah, Akula Ravi Kumar, Boddupally Peda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aaramadaka Sunil Kumar Reddy and Upadhyayula Surya Narayana Murty


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A Screening Method for Potential Anti-Pancreatic Cancer Candidate Compounds Based on Hsp90-Cdc37 Interaction Model in vitro


Hai Zhang, Sen Sun, Qingshan Chen, Guoqing Zhang, Zhenqing Zhang, Duxin Sun and Wenpeng Zhang


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Identification of Novel GSK1070916 Analogs as Potential Aurora B Inhibitors: Insights from Molecular Dynamics and MM/GBSA based Rescoring


Faraz Shaikh, Soumendranath Bhakat, Abhishek Thakur, Ashish Radadia, Mahmoud E. S. Soliman and Anamik Shah


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Synthesis and Analgesic Activity of 3, 7-Dimethylpurine-2, 6-Dion-1-yl Derivatives of Acetic and Butanoic Acid


Malgorzata Zygmunt, Pawel Zmudzki, Grazyna Chlon-Rzepa, Jacek Sapaa and Maciej Pawlowski


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Pd/C-Mediated Synthesis of 3-Methyleneisoindolin-1-ones: Biological and Theoretical Study of their PDE4 Inhibition


Suryadevara Vijayavardhini, Dandela Rambabu, Vegendla Radha, Ravikumar Kapavarapu, Mandava Venkata Basaveswara Rao and Manojit Pal


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Synthesis and Evaluation of Bis-pyrazolineDerivatives as Potential Antimicrobial Agents


Mehlika Dilek Altıntop, Usama Abu Mohsen, Hulya Karaca, Zerrin Cantürk and Ahmet Ozdemir


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Design, Synthesis and in vitro Cytotoxicity Evaluation of new 3', 4'-bis (3, 4, 5-Trisubstituted)-4'H-Spiro [Indene-2, 5'-Isoxazol]-1(3H)-one Derivatives as Promising Anticancer Agents


Hoda Abolhasani, Afshin Zarghi, Ahmad Abolhasani, Maryam Hamzeh-Mivehroud, Nasrin Bargahi, Behrouz Notash, Javid Shahbazi Mojarrad and Siavoush Dastmalchi


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In Vitro and In Vivo Investigations into the Carbene Copper Bromide Anticancer Drug Candidate WBC4

, 2014 :11(7); 825 - 832

Wolfgang Walther, Iduna Fichtner, Frauke Hackenberg, Wojciech Streciwilk and Matthias Tacke


DOI: 10.2174/1570180811666140529004102
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Analysis of Proteasome Inhibition Prediction Using Atom-Based Quadratic Indices Enhanced by Machine Learning Classification Techniques

, 2014 :11(6); 705 - 711

Gerardo M. Casanola-Martin, Huong Le-Thi-Thu, Yovani Marrero-Ponce, Juan A Castillo- Garit, Francisco Torrens, Facundo Perez-Gimenez and Concepcion Abad


DOI: 10.2174/1570180811666140122001144
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Potent Neuroprotective Activity of Monoterpene Derived 4-[(3aR,7aS)- 1,3,3a,4,5,7a-Hexahydro-3,3,6-trimethylisobenzofuran-1-yl]-2-methoxyphenol in MPTP Mice Model

, 2014 :11(5); 611 - 617

Alla V. Pavlova, Irina V. Il'ina, Ekaterina A. Morozova, Dina V. Korchagina, Svetlana Yu. Kurbakova, Irina V. Sorokina, Tatyana G. Tolstikova, Konstantin P. Volcho and Nariman F. Salakhutdinov


DOI: 10.2174/1570180811666131210000316
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Synthesis and Anti-Proliferative Activity of New Biphenyle-Benzylidenethiazolidine- 2,4-dione Bis-Adducts Containing Various Heterocyclic Cores

, 2014 :11(3); 256 - 264

Maxime Meyer, Sandra Kuntz, Isabelle Grillier-Vuissoz, Helene Martin, Lysiane Richert, Stephane Flament, Yves Chapleur and Michel Boisbrun


DOI: 10.2174/15701808113106660080
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Biochemical Changes Evidenced in Alzheimer's Disease: A Mini-Review

, 2014 :11(2); 240 - 248

Luciana Scotti, Francisco Jaime Bezerra Mendonça Junior, Marcelo Sobral da Silva, Ivan R. Pitta and Marcus Tullius Scotti


DOI: 10.2174/15701808113109990063
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