E-Pub Articles Ahead of Print ::: Medicinal Chemistry

ISSN: 1875-6638 (Online)
ISSN: 1573-4064 (Print)


Volume 12, 8 Issues, 2016


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Medicinal Chemistry

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Editor-in-Chief:
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Kings College
University of Cambridge
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Email: mc@benthamscience.org

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E-Pub Articles Ahead of Print

Antimicrobial activity of new 2-Thioxo-benzo[g]quinazolin-4(3H)-one derivatives


Rashad Al-Salahi, Hatem A. Abuelizz, Rabab El Dib and Mohamed Marzouk.


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Benzoflavonoids Structure Hinders Human Colon Cancer Clonogenicity


Yeonjoong Yong, Eun Jee Koh, Seunghyun Ahn, Beom Soo Kim, Young Lee, Soon Young Shin and Yoongho Lim.


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Synthesis and Antifungal Activity of Some 4,6-Dimethylisoxazolo[3,4-b]pyridin-3(1H)-one Derivatives


Jarosław Sączewski, Joanna Fedorowicz, Anna Kędzia, Marta Ziółkowska-Klinkosz and Aleksandra Jalińska.


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Cystic Fibrosis Revisited - a Review Study


Blanka Klimova, Kamil Kuca, Michal Novotny and Petra Maresova.


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Non-Imidazole Histamine H3 Ligands. Part VI. Synthesis and Preliminary Pharmacological Investigation of Thiazole-Type Histamine H3-Receptor Antagonists with Lacking a Nitrogen Nucleus in the Side Chain


Roman Guryn, Marek Staszewski, Piotr Kopczacki and Krzysztof Walczyński.


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An Evaluation on Different Machine Learning Algorithms for Classification and Prediction of Antifungal Peptides


Maryam Mousavizadegan and Hassan Mohabatkar.


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Synthesis and Biological Activities of Lanthanide (III) Nitrate Complexes with N-(2-hydroxynaphthalen-1-yl) methylene) Nicotinohydrazide Schiff Base


Ahmed K. Hijazi, Ziyad A. Taha, Abdulaziz M. Ajlouni, Waleed M. Al-Momani, Idris M. Idris and Eman Abu Hamra.


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Design, Synthesis and Qualitative Structure Activity Relationship Evaluations of Quinoline-Based Bisarylimidazoles as Antibacterial Motifs


Raed A. Al-Qawasmeh, Basil Bani Huthail, Mutasem O. Sinnokrot, Mohammad H. Semreen, Raed Abu Odeh, Musa H. Abu-Zarga, Hamadeh Tarazi, Imad Abu Yousef and Taleb H Al-Tel.


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New Hopes in Cancer Battle - A Review of New Molecules and Treatment Strategies


Marika Turek, Magdalena Krzyczmonik and Piotr Bałczewski.


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Synthesis and Biological Evaluations of Cytotoxic and Antiangiogenic Triterpenoids-Jacaranone Conjugates


Hua Sun, Partick Y. K. Yue, Shao-Rong Wang, Lihong Huo, Ying Zhao, Songbo Xie, Jens Vindahl Kringelum, Ole Lund, Olivier Taboureau, Jun Zhou, Ricky N. S. Wong and Wei-Shuo Fang.


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THREE ARACHIDONOYLAMIDE DERIVATIVES INHIBIT PRO-INFLAMMATORY GENES EXPRESSION BY MODULATING NF-κB AND AP1 ACTIVITIES


Alex Gregorelli, Anna Sgarbossa, Shahbaz Khan, Annunziata Soriente, Margherita De Rosa, Carmela Saturnino and Marta Menegazzi.


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Synergistic Effect of the Combination of Novel Suberoylanilide Hydroxamic Acid Derivatives with Cisplatin on Anti-proliferation of Human Cancer Cells


Rui Xie, Jinghua Shi, Chunhui Cheng, Fan Yun, Xia Liu, Pingwah Tang, Xinying Wu, Ming Yang and Qipeng Yuan.


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Integrated In Silico-In Vitro Discovery of Lung Cancer-related Tumor Pyruvate Kinase M2 (PKM2) Inhibitors


Xiangyun Ye, Yinjia Sun, Yunhua Xu, Zhiwei Chen and Shun Lu.


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Synthesis of cyclic imides (methylphtalimides, carboxylic acid phtalimides and itaconimides) and evaluation of their antifungal potential


Dorimar Stiz, Rogério Corrêa, Felicia Diodata D'Auria, Giovanna Simonetti and Valdir Cechinel-Filho.


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cis-2-Alkenoic acids as promising drugs for the control of biofilm infections


Kamila Tomoko Yuyama and Wolf-Rainer Abraham.


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Synthesis, Anticlotting and Antiplatelet Effects of 1,2,3-Triazoles Derivatives


Laura de Andrade Moura, Ana Carolina Marqui de Almeida, Andreza Vieira da Silva, Vivian Rodrigues de Souza, Vitor Francisco Ferreira, Michel Vieira Menezes, Carlos Roland Kaiser, Sabrina Baptista Ferreira and André Lopes Fuly.


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Microwave Assisted Organic Synthesis of Heterocycles in Aqueous Media: Recent Advances in Medicinal Chemistry


Francesco Frecentese, Irene Saccone, Giuseppe Caliendo, Angela Corvino, Ferdinando Fiorino, Elisa Magli, Elisa Perissutti, Beatrice Severino and Vincenzo Santagada.


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Antimicrobial Activity of Synthesized 2-Methylthiobenzo[g][1,2,4]-triazolo[1,5-a]quinazoline Derivatives


Rashad Al-Salahi, Hatem A. Abuelizz, Mahasin Wadi, Rabab A. El Dib and Mohamed Marzouk.


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Synthesis, Cytotoxic Activity on Leukemia Cell Lines and Quantitative Structure-Activity Relationships (QSAR) Studies of Morita-Baylis-Hillman Adducts


Claudio G. Lima–Junior, Gláucia V. Faheina–Martins, Caio C. B. Bomfim, Everton P. Silva, Demetrius A. M. de Araújo, Edilson B. Alencar Filho and Mário L A A Vasconcellos.


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Synthesis of 1,4-disubstituted 1,2,3-triazole Derivatives Using Click Chemistry and their Src Kinase Activities


Alexandre Lebeau, Cyril Abrioux, David Bénimèlis, Zohra Benfodda and Patrick Meffre.


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Synthesis and Biological Evaluation of N-Aryl-N’-(5-(2-hydroxybenzoyl)pyrimidin-2-yl)guanidines as Toll-Like Receptor 4 Antagonists Synthesis of Guanidine-Based TLR4 Antagonists


Matej Sova, Kaja Rožman, Urban Švajger, Primož Rožman and Stanislav Gobec.


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Facing Chagas’ Disease: Trypanocidal Properties of New Coumarinchalcone Scaffolds


Saleta Vazquez-Rodriguez, Roberto Figueroa Guíñez, Maria João Matos, Claudio Olea-Azar, Juan Diego Maya, Eugenio Uriarte and Lourdes Santana.


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Nitazoxanide Analogues as Antimicrobial Agents Against Nosocomial Pathogens


Jia-Suey Gau, Wen-Pao Lin, Li-Ching Kuo and Ming-Kuan Hu.


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Synthesis, in vivo Anticoagulant Evaluation and Molecular Docking Studies of Bicoumarins Obtained from Furocoumarin Peucedanin


Alla V. Lipeeva, Mikhail V. Khvostov, Dmitry S. Baev, Makhmut M. Shakirov, Tatijana G. Tolstikova and Elvira E Shults.


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Biologically Active New N, N', N''-Tri-Substituted Ferrocenyl Phenylguanidines and their Characterization


Rukhsana Gul, Ataf Ali Altaf, Azim Khan, Amin Badshah, Afzal Shah, Zia ur Rehman, Rabia Naz, Muhammad Nawaz Tahir and Asif Junaid.


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Synthesis and Evaluation of Phenyliminoindolin-Containing Phenylacetamide Derivatives with the Antidepressant and Anticonvulsant Effects


Li-Ping Guan, Bing-Yu Liu, Ying-Chun Quan, Li-Ye Yang, Xing-Hua Zhen and Si-Hong Wang.


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Synthesis, Antibacterial Activity, Interaction with Nucleobase and Molecular Docking Studies of 4-Formylbenzoic Acid Based Thiazoles


Krzysztof Z. Łączkowski, Anna Biernasiuk, Angelika Baranowska-Łączkowska, Konrad Misiura, Anna Malm, Tomasz Plech and Agata Paneth.


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Ether and Carbamate Derivatives of 3-quinuclidinol and 3- hydroxymethylquinuclidine: Synthesis and Evaluation as Nicotinic Ligands


Sivakumar Annadurai, Min Zhang, Jerome L. Gabriel, Merouane Bencheriff and Daniel J Canney.


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Efficient Synthesis and Discovery of Schiff Bases as Potent Cholinesterase Inhibitors


Basma M. Abd Razik, Hasnah Osman, Mohammed Oday Ezzat, Alireza Basiri, Abdussalam Salhin, Yalda Kia and Vikneswaran Murugaiyah.


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Cell-based Assays for Assessing Toxicity: A Basic Guide


Raveen Parboosing, Gugulethu Mzobe, Louis Chonco and Indres Moodley.


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Fluorescein-labeled Bacitracin and Daptomycin Conjugates: Synthesis, Fluorescence Imaging and Evaluation


Sumbla Sheikh, Alexander Sturzu, Hubert Kalbacher, Thomas Nägele, Christopher Weidenmaier, Marius Horger, Christian Schwentner, Ulrike Ernemann and Stefan Heckl.


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Antiplasmodial Limonoids from Trichilia rubescens (Meliaceae)


Tsamo Tontsa Armelle, Nangmo Kemda Pamela, Mkounga Pierre, Ingrid B. Müller, Kirk Marat, Gabriele Sass and Nkengfack Augustin Ephrem.


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Design, Synthesis, and Cytotoxicity of Novel 2,4,6-Trisubstituted 1,3,5- triazines Bearing Aryl Hydrazone Moiety as Potent Antitumor Agent


Limei Wang, Sijia Zhao, Guanglong Bao, Yu Zhang, Shuancheng Xi, Guolin Zhou, Xin Zhai and Ping Gong.


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Synthesis, Biological Evaluation and Pharmacokinetic Studies of Mefenamic Acid - N-Hydroxymethylsuccinimide Ester Prodrug as Safer NSAID


Asif Husain, Priyanka Ahuja, Aftab Ahmad and Shah Alam Khan.


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Robust Modeling and Scaffold Hopping: Case Study Based on HIV Reverse Transcriptase Inhibitors Type-1 Data


Girinath G. Pillai, Laznier Mederos, Chandramukhi S. Panda, Amber Gronski, Peeter Burk, C. Dennis Hall, Alan R. Katritzky, Kaido Tämm and Mati Karelson.


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The Brain Protective Effect of rTMS (Repetitive Transcranial Magnetic Stimulation) in Depression: A Mini-Review in Animal Studies


Burak Yulug, Lütfü Hanoglu, Ahmet Mithat Tavli, Nesrin Helvacı Yılmaz and Ertugrul Kılıc.


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QSRR and QSAR Studies of Antitumor Drugs in View of their Biological Activity Prediction


Paulina Szatkowska-Wandas, Marcin Koba, Grzegorz Smoliński and Jacek Wandas.


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Synthesis and Biological Evaluation of Novel 1,3,4-thiadiazole Derivatives Incorporating Benzisoselenazolone Scaffold as Potential Antitumor Agents


Xiaoyun Fu, Sha Li, Fen Jing, Xuefeng Wang, Baolin Li, Jijun Zhao, Yuming Liu and Baoquan Chen.


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Understanding the Structural Basis of ALDH-2 Inhibition by Molecular Docking


Thayssa T. S. C. Ferreira and Carlos Alberto Manssour Fraga.


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Current medical treatment of early breast cancer


Franco Lumachi.


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