E-Pub Articles Ahead of Print ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 13, 10 Issues, 2016


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Letters in Drug Design & Discovery

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Editor-in-Chief:
Atta-ur-Rahman, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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E-Pub Articles Ahead of Print

Synthesis and Biological Evaluation of Macamides Derivatives as Potent Inhibitors of Breast Cancer Cell MCF-7


Xiao Xia Liang, Cheng Xiong, Min He, Changliang He and Zhongqiong Yin.


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Preparation and Characterization of CS/(β-CD)/PAA Composite Hydrogels for Controlled Drug Delivery


Jie Ren, Xiaoci Yang, Mengqi Yao, Jinfen Gu, Xiaohua Tang and Wu Yang.


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Synthesis and Evaluation of Certain Symmetrical Schiff Bases as Inhibitors of MDA-MB-241 Human Breast Cancer Cell Proliferation


Smaail Radi, Said Tighadouini, Olivier Feron, Olivier Riant and Yahia N Mabkhot LCAE.


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Substituted 1,2,4-oxodiazoles as Potent Inhibitors of Human 11β - hydroxysteroid Dehydrogenase Type 1 (11β-HSD1): Virtual Screening and Docking Results


Dmitry V. Ziolkovskiy, Victoria V. Lipson, Anastasia D. Nikitina and Valentin A Chebanov.


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Design, Synthesis and Biological Evaluation of Salicylamide Analogues as Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitors


Yang Liu, Yijing Li, Jianzhen Liu, Limin Yang, Pengzhan Li and Guisen Zhao.


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Synthesis and Biological Activity of Novel N-Glucosides Containing Substituted Piperazine Moiety


Li-Yuan Zhang, Bao-Lei Wang, Yi-Zhou Zhan, Xue-Wen Hua, Ming Liu, Xiao Zhang, Hai-Bin Song and Zheng-Ming Li.


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Synthesis of Novel C3-Linked β-Carboline-Pyridine Derivatives Employing Khronke Reaction: DNA-binding Ability and Molecular Modeling Studies


Nagula Shankaraiah, Pankaj Sharma, Srinivas Pedapati, Shalini Nekkanti, Vunnam Srinivasulu, Niggula Praveen Kumar and Ahmed Kamal.


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Design, Synthesis and ex vivo Study of the Vasorelaxant Activity Induced by Isosteric Derivatives of Dihydropyridines(NH→O)


Priscila Rendón-Vallejo, Samuel Estrada-Soto, Miguel A. Vázquez, Fernando Hernández-Borja, Rafael Villalobos-Molina and Maximiliano Ibarra-Barajas.


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Synthesis and Antitumor Activity of Novel N-Benzoyl-N'-substituted Pyrimidinyl (Thio)semicarbazide Derivatives


Gaopeng Song, Jianzuo Li, Hao Tian, Yasheng Li, Dekun Hu, Ying Li and Zining Cui.


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Antipsychotics as Psychosis Drugs and Neuroprotective Promoters Evaluated by Chemical QSAR - in silico and in vivo Studies


Maria Mernea, Livia-Cristina Borcan, Florin Borcan and Speranta Avram.


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Flavonoids as Natural Inhibitors of Jack Bean Urease Enzyme


Jalaluddin A. J. Awllia, Maryam AL-Ghamdi, Etimad Huwait, Sumaira Javaid, Atia-tul-Wahab, Saima Rasheed and M Iqbal Choudhary.


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Study of Binding Epitopes by STD-NMR Spectroscopy and Molecular Docking of Urease Inhibitors from Lichens


Vinitha Moolchand Thadhani, Ajmal Khan, Atia-tul-Wahab, Sumaira Javaid, Amsal Shafqat, Zaheer-ul-Haq and M Iqbal Choudhary.


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Potent and Orally Bioavailable Antiplatelet Agent, PLD-301, with the Potential of Overcoming Clopidogrel Resistance


Jingyu Chen and Michael Zhiyan Wang.


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Virtual Screening of NCI Diversity Set IILead to New Cyclin-Dependent Kinases 5Inhibitors Using AutoDock


Siripit Pitchuanchom, Chavi Yenjai, Chantana Boonyarat, Stefano Forli and Arthur J Olson.


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Assembly of Quinoline, Triazole and Oxime Ether in a Single Molecular Entity: A Greener and One-pot Synthesis of Novel Oximes as Potential Cytotoxic Agents


Koduru Sri Shanthi Praveena, Edupuganti Veera Venkat Shivaji Ramarao, Yedia Poornachandra, Chityala Ganesh Kumar, Nallapati Sureshbabu, Nandula Yadagiri Sreenivasa Murthy and Sarbani Pal.


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Peptide Drugs QSAR Modeling Based on a New Descriptor of Amino Acids- SVGT


Jianbo Tong, Lingxiao Li, Shuling Liu and Jia Chang.


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Synthesis and Properties of Brassinosteroid Biosynthesis Inhibitor Fluorescent Probe with Dansyl Moiety


Tomoki Hoshi, Yuko Yoshizawa and Keimei Oh.


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Privileged 1,2,4-Oxadiazoles in Anticancer Drug Design: Novel 5- Aryloxymethyl-1,2,4-oxadiazole Leads for Prostate Cancer Therapy


Alexey Lukin, Ruben Karapetian, Yan Ivanenkov and Mikhail Krasavin.


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Synthesis, Antitumor of New Pyrimidineand Caffeine Derivatives


Ameen Ali Abu-Hashem and Hoda Abdel Raouf Hussein.


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Design, Synthesis and AntitumorActivities of Bis-arylureas and Bisarylamides Based on 1H-benzo[d]imidazole Moiety as Novel BRaf V600E/VEGFR2 Dual Inhibitors


Weimin Yang, Yadong Chen, Yanmin Zhang, Sanzhi Tang, Hongli Chen, Weifang Tang and Tao Lu.


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Synthesis and Biological Activity of Thiazole Dithiocarbamate Derivatives


Nalan Gundogdu-Karaburun.


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Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives


Nalan Gundogdu-Karaburun, Ahmet Cagri Karaburun, Seref Demirayak, Ismail Kayagil and Leyla Yurttas.


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Synthesis and Biological Evaluation of New Tubulin Inhibitors: Shikonin Thio-glycoside Derivatives


Xiao-Ming Wang, Hong-Yan Lin, Jin-Liang Qi, Li-Fei Bai and Yong-Hua Yang.


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Fat-Soluble Vitamins Release Based on Clinoptilolite Zeolite as an Oral Drug Delivery System


Mehdi Rahimi, Hamid Mobedi, Aliasghar Behnamghader, Alireza Nateghi Baygi, Houri Mivehchi and Esmaeil Biazar.


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Synthesis and Biological Evaluations of 3-Benzothiazol-2-yl Coumarin Derivatives as MEK1 Inhibitors


Chao Wang, Fengrong Xu, Yan Niu, Yun Wu, Jing Sun, Yihong Peng, Lei Liang and Ping Xu.


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Synthesis and Biological Evaluation of Arylthiourea Derivatives with Antitubercular Activity


Rusong Luo, Tuomo Laitinen, Liyan Teng, Tapio Nevalainen, Maija Lahtela-Kakkonen, Baofu Zheng, Honghai Wang, Antti Poso and Xuelian Zhang.


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Synthesis and Antiproliferative Evaluation of Hybrids of Indolin-2-one and Quinazoline-4(3H)-one Linked via Imine Bond


Wei-Yao Wu, Sheng-Li Cao, Bei-Bei Mao, Ji Liao, Zhong-Feng Li, Hao-Bin Song and Xingzhi Xu.


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Construction and High Expression of a Recombinant Amino-Proximal HSV-2 Glycoprotein B Polypeptide with Immunogenicity in Escherichia coli


Xu Ning, Tu Jingjing, Wang Xian Yan and Xu Fang.


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Synthesis and Study of Antitumor Activity of Artimisinin Glucoside


Yanrong Ren and Guoping Chen.


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Synthesis and Biological Activity of New 2,3-dihydro-1H-cyclopenta[b]- quinoline Derivatives as Acetylcholinesterase Inhibitors


Pawel Szymanski, Magdalena Markowicz, Marek Bajda, Barbara Malawska and Elzbieta Mikiciuk-Olasik.


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Novel Aminoalcohol Derivatives Bearing 4-Phenylphenol as Antischistosomal Drugs


Li-Ping Duan, Jian Xue, Yi Tao and Hao-Bing Zhang.


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Deformable Surfactant Vesicles Loading Ammonium Glycyrrhizinate: Characterization and In Vitro Permeation Studies


Luisa Di Marzio, Carlotta Marianecci, Federica Rinaldi, Sara Esposito and Maria Carafa.


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