E-Pub Articles Ahead of Print ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 13, 10 Issues, 2016


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Letters in Drug Design & Discovery

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Editor-in-Chief:
Atta-ur-Rahman, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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E-Pub Articles Ahead of Print

Design And Evaluation of Microwave Induced Solid Dispersion of Tinidazole and Molecular Modelling with β-cyclodextrin


Swati Jagdale, Anish Kulkarni, Anuruddha Chabukswar and Bhanudas Kuchekar.


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Synthesis and Antiproliferative Activity of 2-arylidene 6-(2-aryl-2- oxoethoxy)Benzofuran-3-one Derivatives


Seref Demirayak, Leyla Yurttas, Ahmet Cagri Karaburun, Nalan Gundogdu-Karaburun and Ismail Kayagil.


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Arginine-rich Cyclic Peptides Enhance Cellular Delivery of Anticancer Agents: Molecular Insights


Antara Banerjee, Naser Sayeh, Amir Nasrolahi Shirazi, Rakesh Tiwari, Keykavous Parang and Arpita Yadav.


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Effect of Substituted Benzimidazoles and Somatostatin Analogs on the Vitality of Tumor Cell Lines and on the Oxidative Burst of Phagocytes


Ivan Goshev, Emilia Naydenova, Svetlana Staykova, Anelia Mavrova, Ljubomir Vezenkov and Diana Wesselinova.


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In silico Strategies to Probe Stereoselective Interactions of Multidrug Resistant Transporter P-glycoprotein


Ishrat Jabeen.


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Novel Biphenyl Derivatives with α-Aminophosphonate Moiety: Design, Synthesis and Antivirus Activity


Guo Ping Zhang.


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Pharmacokinetics of Selegiline in a Rabbit Model


Huba Kalasz.


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Cytotoxicity of Hydrazones of Morpholine Bearing Mannich Bases towards Huh7 and T47D Cell lines and Their Effects on Mitochondrial Respiration


Kaan Kucukoglu, Halise Inci Gul, Mustafa Gul, Rengul Cetin-Atalay, Yosra Baratli and Bernard Geny.


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Synthesis of Some Novel 2-Azetidinones/4-Thiazolidinones Bearing 1, 3, 4-Thiadiazole Nucleus and Screening for Its Anti-Imflammatory Activity


B. Gowramma, T. K. Praveenc, R. Kalirajana and B Babub.


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Synthesis and Biological Evaluation of Some New Indolizine Derivatives as Antitumoral Agents


Liliana Lucescu, Elena Bicu, Dalila Belei, Joelle Dubois and Alina Ghinet.


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Synthesis and Anticonvulsant Activity of Novel 3-(2-(4H-1,2,4-triazol-4-yl)ethyl)-1-alkyl-1H-indole Derivatives


Zhe-Shan Quan.


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An Efficient Nonconventional Glycerol-Based Solid Acid Catalyzed Synthesis and Biological Evaluation of Phosphonate Conjugates of 1,2,4-Triazole Thiones


M SR Murty.


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Synthesis of 2-, 3- or 4-Phenylsubtituted Chalcones Based on 4-Phenylamino-6-Nitro-2-[(E)-2-Phenylvinyl] Quinoline, Evaluation of their Antimicrobial and Antifungal Activity


Sulochna Mudaliyar, Kishor H. Chikhalia and Nisha K Shah.


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Synthesis and Anticancer Activity of 2-Aryl-6-diethylaminoquinazolinone Derivatives


Won-Jea Cho and Thanh Nguyen Lea.


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Preparation of Chlorotoxin-conjugated Superparamagnetic Nanoparticle and its Magnetic Resonance Imaging In Vitro


Chen Zhu, Xiao Enhua, Shang Quanliang, Kang Zhen, Tan Huilong, Pengfei Xu and Zeng Wenbin.


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Synthesis and Biological Evaluation of Macamides Derivatives as Potent Inhibitors of Breast Cancer Cell MCF-7


Xiao Xia Liang, Cheng Xiong, Min He, Changliang He and Zhongqiong Yin.


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Preparation and Characterization of CS/(β-CD)/PAA Composite Hydrogels for Controlled Drug Delivery


Jie Ren, Xiaoci Yang, Mengqi Yao, Jinfen Gu, Xiaohua Tang and Wu Yang.


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Substituted 1,2,4-oxodiazoles as Potent Inhibitors of Human 11β - hydroxysteroid Dehydrogenase Type 1 (11β-HSD1): Virtual Screening and Docking Results


Dmitry V. Ziolkovskiy, Victoria V. Lipson, Anastasia D. Nikitina and Valentin A Chebanov.


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Synthesis of Novel C3-Linked β-Carboline-Pyridine Derivatives Employing Khronke Reaction: DNA-binding Ability and Molecular Modeling Studies


Nagula Shankaraiah, Pankaj Sharma, Srinivas Pedapati, Shalini Nekkanti, Vunnam Srinivasulu, Niggula Praveen Kumar and Ahmed Kamal.


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Synthesis, Antitumor of New Pyrimidineand Caffeine Derivatives


Ameen Ali Abu-Hashem and Hoda Abdel Raouf Hussein.


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Design, Synthesis and AntitumorActivities of Bis-arylureas and Bisarylamides Based on 1H-benzo[d]imidazole Moiety as Novel BRaf V600E/VEGFR2 Dual Inhibitors


Weimin Yang, Yadong Chen, Yanmin Zhang, Sanzhi Tang, Hongli Chen, Weifang Tang and Tao Lu.


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Synthesis and Biological Activity of Thiazole Dithiocarbamate Derivatives


Nalan Gundogdu-Karaburun.


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Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives


Nalan Gundogdu-Karaburun, Ahmet Cagri Karaburun, Seref Demirayak, Ismail Kayagil and Leyla Yurttas.


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Synthesis and Biological Evaluation of New Tubulin Inhibitors: Shikonin Thio-glycoside Derivatives


Xiao-Ming Wang, Hong-Yan Lin, Jin-Liang Qi, Li-Fei Bai and Yong-Hua Yang.


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Fat-Soluble Vitamins Release Based on Clinoptilolite Zeolite as an Oral Drug Delivery System


Mehdi Rahimi, Hamid Mobedi, Aliasghar Behnamghader, Alireza Nateghi Baygi, Houri Mivehchi and Esmaeil Biazar.


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Synthesis and Biological Evaluations of 3-Benzothiazol-2-yl Coumarin Derivatives as MEK1 Inhibitors


Chao Wang, Fengrong Xu, Yan Niu, Yun Wu, Jing Sun, Yihong Peng, Lei Liang and Ping Xu.


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Synthesis and Biological Evaluation of Arylthiourea Derivatives with Antitubercular Activity


Rusong Luo, Tuomo Laitinen, Liyan Teng, Tapio Nevalainen, Maija Lahtela-Kakkonen, Baofu Zheng, Honghai Wang, Antti Poso and Xuelian Zhang.


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Synthesis and Antiproliferative Evaluation of Hybrids of Indolin-2-one and Quinazoline-4(3H)-one Linked via Imine Bond


Wei-Yao Wu, Sheng-Li Cao, Bei-Bei Mao, Ji Liao, Zhong-Feng Li, Hao-Bin Song and Xingzhi Xu.


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Construction and High Expression of a Recombinant Amino-Proximal HSV-2 Glycoprotein B Polypeptide with Immunogenicity in Escherichia coli


Xu Ning, Tu Jingjing, Wang Xian Yan and Xu Fang.


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Synthesis and Study of Antitumor Activity of Artimisinin Glucoside


Yanrong Ren and Guoping Chen.


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Synthesis and Biological Activity of New 2,3-dihydro-1H-cyclopenta[b]- quinoline Derivatives as Acetylcholinesterase Inhibitors


Pawel Szymanski, Magdalena Markowicz, Marek Bajda, Barbara Malawska and Elzbieta Mikiciuk-Olasik.


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Novel Aminoalcohol Derivatives Bearing 4-Phenylphenol as Antischistosomal Drugs


Li-Ping Duan, Jian Xue, Yi Tao and Hao-Bing Zhang.


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Deformable Surfactant Vesicles Loading Ammonium Glycyrrhizinate: Characterization and In Vitro Permeation Studies


Luisa Di Marzio, Carlotta Marianecci, Federica Rinaldi, Sara Esposito and Maria Carafa.


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